| 常用名 | A-381393 | CAS号 | 726174-00-1 |
|---|---|---|---|
| 价格 | ¥需询单/1g ¥需询单/1mg | 纯度 | 98.0% |
| 备货期 | 需询单 | 库存 | 询单 |
| 产品详情(用途,包装等)
用途: A-381393 is a potent, selective, brain penetrate dopamine D4 receptor antagonist, with Kis of 1.5, 1.9 and 1.6 nM for human dopamine D4.4, D4.2, and D4.7 receptor, respectively, >2700-fold selectivity over D1, D2, D3 and D5 dopamine receptors. A-381393 shows moderate affinity for 5-HT2A (Ki, 370 nM)[1]. 物理化学性质: CAS号:726174-00-1 常用中文名:A-381393 常用英文名:A-381393 分子式:C20H24N4 分子量:320.43 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A 储存条件:2-8℃ |