CGP25454A
更新时间：2026-01-16 21:07:42
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| 常用名 | CGP 25454A | CAS号 | 104391-26-6 |
|---|---|---|---|
| 价格 | 纯度 | 99.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情（用途，包装等）
用途： CGP 25454A is a novel and selective presynaptic dopamine autoreceptor antagonist. In vitro: CGP 25454A increase the field-stimulated [3H]- and [14C]-overflow from rat striatal slices preloaded with [3H]dopamine and [14C]choline, indicating that CGP 25454A is able to enhance the release of both dopamine (DA) and acetylcholine (ACh). However, CGP 25454A is 12.9 times more potent in increasing, by 1/6 of the apparent maximal increase, the release of [3H]DA than that of [14C]ACh.In vivo: CGP 25454A increase [3H]spiperone binding to receptors of the D2 family in rat striatum by 90-110% (ED50: 13 mg/kg i.p.). As a similar increase in [3H]spiperone binding is found with a variety of agents which increase the synaptic concentration of endogenous DA, the effect of CGP 25454A most probably reflects an enhanced release of DA under in vivo conditions. At 30-100 mg/kg, CGP 25454A inhibit [3H]spiperone binding in the pituitary of the same animals as a result of a blockade of postsynaptic DA receptors. 物理化学性质： CAS号：104391-26-6 常用中文名：CGP 25454A 常用英文名：CGP 25454A 分子式：C15H21Cl2N3O2 分子量：346.252 密度：N/A 沸点：N/A 熔点：N/A 闪点：N/A 储存条件：2-8℃ |
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- 产品名：CGP 25454A
- 价格： ￥16500.9/100mg ￥2800.9/5mg ￥4800.9/10mg ￥9600.9/50mg
- 纯度：99.0%
- 备货期：10天
- 联系人：阿拉丁
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参考价格：$320/10mM*1mLinDMSO