| 常用名 | NF157 | CAS号 | 104869-26-3 |
|---|---|---|---|
| 价格 | 纯度 | 98.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: NF157 is a highly selective nanomolar P2Y11 antagonist with a pKi of 7.35. The IC50s are 463 nM, 1811 µM, 170 µM for P2Y11 (Ki=44.3 nM), P2Y1 (Ki=187 µM), P2Y2 (Ki=28.9 µM), respectively. NF157, significantly reduces expression of metalloproteinase (MMP)-3, MMP-13, can be used in the treatment of osteoarthritis (OA). 物理化学性质: CAS号:104869-26-3 常用中文名:NF157 常用英文名:NF 157 分子式:C49H28F2N6Na6O23S6 分子量:1437.10000 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A |