| 常用名 | (S)-(+)-Dimethindene maleate | CAS号 | 136152-65-3 |
|---|---|---|---|
| 价格 | 纯度 | 99.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: (S)-(+)-Dimethindene maleate, an enantiomer, is a potent M2-selective muscarinic receptor antagonist (pA2 = 7.86/7.74; pKi = 7.78). (S)-(+)-Dimethindene maleate shows lower affinities for the muscarinic M1 (pA2 = 6.83/6.36; pKi = 7.08), the M3 (pA2 = 6.92/6.96; pKi = 6.70) and the M4 receptors (pKi = 7.00), respectively. (S)-(+)-Dimethindene maleate also is a histamine H1 receptor antagonist (pA2 = 7.8)[1]. 物理化学性质: CAS号:136152-65-3 常用中文名:(S)-(+)-Dimethindene maleate 常用英文名:(S)-(+)-Dimethindene maleate 分子式:C24H28N2O4 分子量:408.490 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A |