| 常用名 | Bisindolylmaleimide VIII acetate | CAS号 | 138516-31-1 |
|---|---|---|---|
| 价格 | 纯度 | 99.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: Bisindolylmaleimide VIII acetate (Ro 31-7549 acetate) is a potent and selective protein kinase C (PKC) inhibitor with an IC50 of 158 nM for rat brain PKC. Bisindolylmaleimide VIII acetate has IC50s of 53, 195, 163, 213, and 175 nM for PKC-α, PKC-βI, PKC-βII, PKC-γ, PKC-ε, respectively[1]. Bisindolylmaleimide VIII acetate facilitates Fas-mediated apoptosis and inhibits T cell-mediated autoimmune diseases[2]. 物理化学性质: CAS号:138516-31-1 常用中文名:Bisindolylmaleimide VIII acetate 常用英文名:Bisindolylmaleimide VIII acetate 分子式:C26H26N4O4 分子量:458.509 密度:N/A 沸点:693ºC at 760 mmHg 熔点:N/A 闪点:372.9ºC 储存条件:2-8°C,密封,干燥 |