| 常用名 | Dyrk1A-IN-5 | CAS号 | 1685235-41-9 |
|---|---|---|---|
| 价格 | 纯度 | 98.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: Dyrk1A-IN-5 (compound 5j) is a potent and selective DYRK1A inhibitor, with an IC50 of 6 nM. Dyrk1A-IN-5 dose-dependently reduces the phosphorylation of Thr434 in SF3B1, with an IC50 of 0.5 μM. Dyrk1A-IN-5 inhibits phosphorylation of tau at Thr212, with an IC50 of 2.1 μM. Dyrk1A-IN-5 can be used for Down syndrome research[1]. 物理化学性质: CAS号:1685235-41-9 常用中文名:Dyrk1A-IN-5 常用英文名:Dyrk1A-IN-5 分子式:C16H9IN2O2 分子量:388.16 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A |