| 常用名 | (2S,4R)-N-(2-(2-(2-(2-((6-氯己基)氧基)乙氧基)乙氧基)乙氧基)-4-(4-甲基噻唑-5-基)苄基)-1-((S)-2-(1-氰基环丙烷甲酰胺)-3,3-二甲基丁酰基)-4-羟基吡咯烷-2-甲酰胺 | CAS号 | 2365478-58-4 |
|---|---|---|---|
| 价格 | 纯度 | 98.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: HaloPROTAC-E is a novel HaloPROTAC potent degrader, inducing reversible degradation of two endosomally localized proteins, SGK3 and VPS34, with a DC50 of 3-10 nM, remarkably selective inducing only degradation of the Halo tagged endogenous VPS34 complex (VPS34, VPS15, Beclin1, and ATG14). 物理化学性质: CAS号:2365478-58-4 常用中文名:(2S,4R)-N-(2-(2-(2-(2-((6-氯己基)氧基)乙氧基)乙氧基)乙氧基)-4-(4-甲基噻唑-5-基)苄基)-1-((S)-2-(1-氰基环丙烷甲酰胺)-3,3-二甲基丁酰基)-4-羟基吡咯烷-2-甲酰胺 常用英文名:HaloPROTAC-E 分子式:C39H56ClN5O8S 分子量:790.41 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A |