| 常用名 | PFI-2盐酸盐 | CAS号 | 1627607-87-7 |
|---|---|---|---|
| 价格 | 纯度 | 98.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: PFI-2 hydrochloride is a a first-in-class, potent, highly selective, and cell-active inhibitor of the methyltransferase activity of SETD7 with IC50 of 2 nM, 500 fold active than (S)-PFI-2.IC50 value: 2 nM [1]Target: SETD7(R)-PFI-2 is highly selective (>1,000-fold) for SETD7, over a panel of 18 other human protein methyltransferases and DNMT1, and was shown to be inactive against 134 additional ion channel, GPCR, and enzyme targets ( 物理化学性质: CAS号:1627607-87-7 常用中文名:PFI-2盐酸盐 常用英文名:(R)-PFI 2 hydrochloride 分子式:C23H26ClF4N3O3S 分子量:535.982 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A 储存条件:-20℃ |