127785-96-0

• 常用中文名：6-氨甲基-6,11-二氢-5H-二苯并[b,e]氮杂卓富马酸盐
• 常用英文名：6-AMINOMETHYL-6, 11-DIHYDRO-5H-DIBENEZ[B,E]AZEPINE (E)-2-BUTENEDIOATE
• CAS号：127785-96-0
• 分子式：C₁₉H₂₀N₂O₄
• 分子量：340.37300
• 发布时间：2018-12-30 19:06:22
• 更新时间：2026-07-16 18:43:38

名称

• 中文名: 6-氨甲基-6,11-二氢-5H-二苯并[b,e]氮杂卓富马酸盐
• 英文名: (6,11-Dihydro-5H-dibenzo[b,e]azepin-6-yl)methanamine fumarate
• 中文别名: (6,11-二氢-5H-二苯并[B,E]氮杂卓-6-基)甲胺富马酸盐; 依匹斯汀杂质44 富马酸盐; 依匹斯汀杂质8; 依匹斯汀相关化合物A富马酸盐; 依匹斯汀杂质A024-V对照品
• 英文别名: 6,11-dihydro-5H-Dibenz[b,e]azine-6-methanamine (2E)-2-butenedioate (1:1) (9CI ACI); *Prilocaine Impurity 32; 5H-Dibenz[b,e]azine-6-methanamine, 6,11-dihydro-, (2E)-2-butenedioate (1:1) (9CI, ACI); Ethyl 3-[[2-[[4-(N-Hexoxycbonylcbamimidoyl)-N-nitroso-anilino]methyl]-1-methyl-benzimidazole-5-carbonyl]-(2-pyridyl)amino]propanoate; 6-AMIOMETHYL-6,11-DIHYDRO-5H-DIBENZ[B,E]AZIN(E)-2-BUTANEDIOATE(1:1); 6-AMINOMETHYL-6,11-DIHYDRO-5H-DIBENZ[B,E]AZINE (E)-2-BUTENEDIOATE; 6-aMinoMethyl-6,11-dihydro-5H-dibenz[b,e]azine succinate; inastine RC A; inastine Impurity A024-V; inastine Related Compound A Fumate; 6-aminomethy,11-dihydro-5H-dibenz[b,e]azine fumate; inastine Impurity 8; 6-Aminomethyl-6,11-dihydro-5H-dibenz[b,e]azepine (E)-2-butenedioate; 6-Aminomethyl-6,11-Dihydro-5H-dibenzo [b, e] azetidine fumate; inastine Impurity 44 Fumate; 6-AMINOMETHYL-6, 11-DIHYDRO-5H-DIBENEZ[B,E]AZINE (E)-2-BUTENEDIOATE; 5H-Dibenz[b,e]azine-6-methanamine, 6,11-dihydro-, (2E)-2-butenedioate (1:1); (6,11-Dihydro-5H-dibenzo[b,e]azin-6-yl)methanamine fumate; inastine hydrochloride intermediate

物化性质

• 沸点: 616.9ºC at 760 mmHg
• 分子式: C₁₉H₂₀N₂O₄
• 分子量: 340.37300
• 闪点: 326.9ºC
• 精确质量: 340.14200
• PSA: 112.65000
• LogP: 3.25280
• 蒸汽压: 4.48E-16mmHg at 25°C
• 储存条件: 室温

安全

• 海关编码: 2933990090

合成路线

74860-00-7 110-17-8 ~76% 127785-96-0

文献：Konica Minolta Chemical Co., Ltd. Patent: EP1496051 A1, 2005 ; Location in patent: Page 3 ;

41218-84-2 110-17-8 ~% 127785-96-0

文献：WO2009/63504 A2, ; Page/Page column 24 ;

上下游产品

上游产品  3
74860-00-7 110-17-8 41218-84-2
下游产品  1
80012-43-7

海关

海关编码	2933990090
中文概述	2933990090. 其他仅含氮杂原子的杂环化合物. 增值税率:17.0%. 退税率:13.0%. 监管条件:无. 最惠国关税:6.5%. 普通关税:20.0%
申报要素	品名, 成分含量, 用途, 乌洛托品请注明外观, 6－己内酰胺请注明外观, 签约日期
Summary	2933990090. heterocyclic compounds with nitrogen hetero-atom(s) only. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:20.0%