中文名 | 阿必鲁泰 |
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英文名 | Albiglutide |
英文别名 |
Gsk 716155
7-36-Glucagon-like peptide I (8-glycine) (human), fusion protein with 7-36-glucagon-like peptide I (8-glycine) (human) fusion protein with serum Albugon Naliglutide Unii-5E7U48495e 7-36-Glucagon-likepeptide I [8-glycine] (huMan), fusion protein with 7-36-glucagon-like peptide I[8-glycine] (huMan) fusion protein with seruM albuMin (huMan) L-Histidylglycyl-L-α-glutamylglycyl-L-threonyl-L-phenylalanyl-L-threonyl-L-seryl-L-α-aspartyl-L-valyl-L-seryl-L-seryl-L-tyrosyl-L-leucyl-L-α-glutamylglycyl-L-glutaminyl-L-alanyl-L-alanyl-L
 -lysyl-L-α-glutamyl-L-phenylalanyl-L-isoleucyl-L-alanyl-L-tryptophyl-L-leucyl-L-valyl-L-lysylglycyl-L-argininamide L-Argininamide, L-histidylglycyl-L-α-glutamylglycyl-L-threonyl-L-phenylalanyl-L-threonyl-L-seryl-L-α-aspartyl-L-valyl-L-seryl-L-seryl-L-tyrosyl-L-leucyl-L-α-glutamylglycyl-L-glutaminyl-L-a
 lanyl-L-alanyl-L-lysyl-L-α-glutamyl-L-phenylalanyl-L-isoleucyl-L-alanyl-L-tryptophyl-L-leucyl-L-valyl-L-lysylglycyl- |
描述 | 阿比鲁肽是一种胰高血糖素样肽-1(GLP-1)模拟物,是一种长效GLP-2受体激动剂。阿比鲁肽显著降低糖化血红蛋白(A1C)。阿比鲁肽可用于2型糖尿病(T2D)研究。阿比鲁肽是由抗DPP-4的GLP-1二聚体与人白蛋白的遗传融合产生的[1][2][3]。 |
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相关类别 | |
参考文献 |
密度 | 1.5±0.1 g/cm3 |
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分子式 | C148H224N40O45 |
分子量 | 3283.603 |
精确质量 | 3281.646973 |
LogP | -5.20 |
外观性状 | 粉末 |
折射率 | 1.661 |
储存条件 | -20℃ |