42399-40-6

• 常用中文名：去乙酰地尔硫卓
• 常用英文名：Deacetyldiltiazem
• CAS号：42399-40-6
• 分子式：C₂₀H₂₄N₂O₃S
• 分子量：372.48100
• 发布时间：2018-07-10 19:08:39
• 更新时间：2026-07-12 20:39:08
• Deacetyldiltiazem is a metabolite product of the drug Diltiazem (a coronary vasodilator), and is present in the plasma of individuals taking that medication.

名称

• 中文名: 去乙酰地尔硫卓
• 英文名: Desacetyl Diltiazem
• 中文别名: 去乙酰地尔硫卓(游离态); 去乙酰地尔硫卓杂质F; 脱乙基地尔硫卓; O-去乙酰地尔硫卓-D6; 盐酸地尔硫卓杂质F; 地尔硫卓 杂质 F(去乙酰地尔硫卓); (2S-cis)-5-(2-(二甲基氨基)乙基)-2,3-二氢-3-羟基-2-(4-甲氧基苯基)-1,5-苯并硫氮杂卓-4(5H)-酮; 盐酸去乙酰地尔硫卓; 盐酸地尔硫卓杂质F 标准品; 去乙酰地尔硫卓/(2S-CIS)-5-(2-(二甲基氨基)乙基)-2,3-二氢-3-羟基-2-(4-甲氧基苯基)-1,5-苯并硫氮杂卓-4(5H)-酮; 盐酸地尔硫杂质Ⅰ(去乙酰地尔硫); O-去乙酰地尔硫卓; 盐酸地尔硫杂质Ⅰ(去乙酰地尔硫)
• 英文别名: Diltiazem Hydrochloride Impurity F; 5-[2-(Dimethylamino)ethyl]-3-hydroxy-2,3-dihydro-2-(4-methoxyphenyl)-1,5-benzothiazin-4(5H)-one; (2S-cis)-5-[2-(dimethylamino)ethyl]-2,3-dihydro-3-hydroxy-2-(4-methoxyphenyl)-1,5-benzothiazin-4(5H)-one; (2s-Cis)-5-((Dimethylamino)Ethyli)-2,3-Dihydro-3-Hydroxy-2-(4-Methoxyphenyl)-1,5-Benzothiazin-4(5h)-One; [2S,(+)]-3β-Hydroxy-5-[2-(dimethylamino)ethyl]-2,3-dihydro-2β-(4-methoxyphenyl)-1,5-benzothiazin-4(5H)-one; Diltiazem Hydrochloride Impurit Ⅰ:Deacetyldiltiazem; Diltiazem Impurity F (Desacetyl Diltiazem); d-cis-Desacetyldiltiazem; (2S,3S)-5-[2-(Dimethylamino)ethyl]-3-hydroxy-2-(4-methoxyphenyl)-2,3-dihydro-1,5-benzothiazin-4(5H; (2S,3S)-5-[2-(Dimethylamino)ethyl]; 3-Hydroxy-5-[2-(dimethylamino)ethyl]-2,3-dihydro-2-(4-methoxyphenyl)-1,5-benzothiazin-4(5H)-one; 1,5-Benzothiazin-4(5H)-one, 5-[2-(dimethylamino)ethyl]-2,3-dihydro-3-hydroxy-2-(4-methoxyphenyl)-, (2S,3S); (2S)-5-[2-(Dimethylamino)ethyl]-2,3-dihydro-3β-hydroxy-2β-(4-methoxyphenyl)-1,5-benzothiazin-4(5H)-one; (2S)-5-[2-(Dimethylamino)ethyl]-2,3-dihydro-3β-hydroxy-2-(4-methoxyphenyl)-1,5-benzothiazin-4(5H)-one; Deacetyldiltiazem hydrochloride; (2S)-2-(4-Methoxyphenyl)-3β-hydroxy-5-[2-(dimethylamino)ethyl]-2,3-dihydro-1,5-benzothiazine-4(5H)-one; Desacetyldiltiazem 1.0 mg/ml in Acetonitrile; DiltiazeM IMpurity F; Desacetyl DiltiazemQ: What is Desacetyl Diltiazem Q: What is the CAS Number of Desacetyl Diltiazem Q: What is the storage condition of Desacetyl Diltiazem Q: What e the applications of Desacetyl Diltiazem; (2S,3S)-2,3-Dihydro-2-(4-methoxyphenyl)-3-hydroxy-5-[2-(dimethylamino)ethyl]-1,5-benzothiazine-4(5H)-one; (3S,4S)-6-(2-dimethylaminoethyl)-4-hydroxy-3-(4-methoxyphenyl)-2-thia-6-azabicyclo[5.4.0]undeca-7,9,11-trien-5-one; Diltiazem Impurity 6 Monomer; (2S-cis)-5-[(Dimethylamino)ethyl]-2,3-dihydro-3-hydroxy-2-(4-methoxyphenyl)-1,5-benzothiazin-4(5H)-one; O-Desacetyl Diltiazem-d6; Deacetyl-d-diltiazem; (2S-cis)-5-(2-(Dimethylamino)ethyl)-2,3-dihydro-3-hydroxy-2-(4-methoxyphenyl)-1,5-benzothiazin-4(5H)-one; Diltiazem-Imp-F; (2S,3S)-5-[2-(Dimethylamino)ethyl]-2-(4-methoxyphenyl)-4-oxo-2,3,4,5-tetrahydro-1,5-benzothiazin-3-ol; (2S,3S)-5-(2-(Dimethylamino)ethyl)-3-hydroxy-2-(4-methoxyphenyl)-2,3-dihydrobenzo[b][1,4]thiazin-4(5H)-one

物化性质

• 密度: 1.225g/cm3
• 沸点: 596.8ºC at 760mmHg
• 分子式: C₂₀H₂₄N₂O₃S
• 分子量: 372.48100
• 闪点: 314.8ºC
• 精确质量: 372.15100
• PSA: 78.31000
• LogP: 2.86270
• 外观性状: 灰白色至淡黄色固体
• 折射率: 1.609

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