Galnon (trifluoroacetate salt)

• 常用名: Galnon (trifluoroacetate salt)
• 英文名: Galnon (trifluoroacetate salt)
• CAS号: 1217448-19-5
• 分子量: 792.840
• 密度: N/A
• 沸点: N/A
• 分子式: C₄₂H₄₇F₃N₄O₈
• 熔点: N/A
• 闪点: N/A

Galnon (trifluoroacetate salt)用途

半乳糖凝集素-TFA是半乳糖凝集素GAL1和GAL2受体的选择性非肽激动剂,Kis分别为11.7和34.1μM。Galnon TFA具有抗惊厥和抗焦虑作用[1][2]。

Galnon (trifluoroacetate salt)名称

• 英文名: Galnon (trifluoroacetate salt)

Galnon (trifluoroacetate salt)生物活性

• 描述: 半乳糖凝集素-TFA是半乳糖凝集素GAL1和GAL2受体的选择性非肽激动剂,Kis分别为11.7和34.1μM。Galnon TFA具有抗惊厥和抗焦虑作用[1][2]。
• 相关类别:
  研究领域 >> 神经疾病
  信号通路 >> G 蛋白偶联受体/G 蛋白 >> 神经肽Y受体
• 参考文献:

  [1]. Bartfai T, et, al. Galmic, a nonpeptide galanin receptor agonist, affects behaviors in seizure, pain, and forced-swim tests. Proc Natl Acad Sci U S A. 2004 Jul 13;101(28):10470-5.

  [2]. Rajarao SJR, et, al. Anxiolytic-like activity of the non-selective galanin receptor agonist, galnon. Neuropeptides. 2007 Oct;41(5):307-20.

Galnon (trifluoroacetate salt)物理化学性质

• 分子式: C₄₂H₄₇F₃N₄O₈
• 分子量: 792.840
• 精确质量: 792.334595

Galnon (trifluoroacetate salt)英文别名

• 3-Cyclohexyl-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-alanyl-N-(4-methyl-2-oxo-2H-chromen-7-yl)-L-lysinamide trifluoroacetate (1:1)
• Galnon (trifluoroacetate salt)
• 7-((9-Fluorenylmethoxycarbonyl)cyclohexylalanyllysyl) amino-4-methylcoumarin trifluoroacetate salt
• MFCD06798339
• Galnon trifluoroacetate salt
• Acetic acid, 2,2,2-trifluoro-, compd. with L-lysinamide, 3-cyclohexyl-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-alanyl-N-(4-methyl-2-oxo-2H-1-benzopyran-7-yl)- (1:1)