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JNJ-56022486

更新时间:2025-07-31 17:03:44

JNJ-56022486结构式
JNJ-56022486结构式
品牌特惠专场
常用名 JNJ-56022486 英文名 JNJ-56022486
CAS号 2036082-79-6 分子量 283.72
密度 N/A 沸点 N/A
分子式 C15H10ClN3O 熔点 N/A
MSDS N/A 闪点 N/A

 JNJ-56022486用途


含TARP-gamma8的AMPA受体新型高效选择性负性调节剂

 JNJ-56022486名称

英文名 JNJ-56022486

 JNJ-56022486生物活性

描述 含TARP-gamma8的AMPA受体新型高效选择性负性调节剂

 JNJ-56022486物理化学性质

分子式 C15H10ClN3O
分子量 283.72

 JNJ-56022486靶点实验

查看更多实验

实验名称:Apparent permeability across apical to basolateral side in MDCK-MDR1 cells at 5 uM me...
来源:ChEMBL
靶标:N/A
External Id:CHEMBL4200551
实验名称:Apparent permeability across basolateral to apical side in MDCK-MDR1 cells at 5 uM me...
来源:ChEMBL
靶标:N/A
External Id:CHEMBL4200550
实验名称:Hepatic extraction ratio in rat liver microsomes at 1 uM measured after 60 mins in pr...
来源:ChEMBL
靶标:N/A
External Id:CHEMBL4200549
实验名称:Hepatic extraction ratio in human liver microsomes at 1 uM measured after 60 mins in ...
来源:ChEMBL
靶标:N/A
External Id:CHEMBL4200548
实验名称:Modulation of recombinant human GluA1 flop isoform/TARPgamma8 expressed in HEK293F ce...
来源:ChEMBL
靶标:Voltage-dependent calcium channel gamma-8 subunit
External Id:CHEMBL4200544
实验名称:Calcium Flux Assay from US Patent US10611730: "Benzimidazolone and benzothiazolone co...
来源:BindingDB
靶标:N/A
External Id:BindingDB_9024_1
实验名称:Protein binding in rat plasma assessed as unbound fraction at 1 uM measured after 6 h...
来源:ChEMBL
靶标:N/A
External Id:CHEMBL4200555
实验名称:Protein binding in human plasma assessed as unbound fraction at 1 uM measured after 6...
来源:ChEMBL
靶标:N/A
External Id:CHEMBL4200554
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