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B-Raf IN 2

更新时间:2025-08-27 11:33:07

B-Raf IN 2结构式
B-Raf IN 2结构式
品牌特惠专场
常用名 B-Raf IN 2 英文名 B-Raf IN 2
CAS号 2649372-20-1 分子量 461.44
密度 N/A 沸点 N/A
分子式 C20H17F2N5O4S 熔点 N/A
MSDS N/A 闪点 N/A

 B-Raf IN 2用途


B-Raf IN 2是一种有效的选择性BRAF抑制剂,从专利WO2021116055A1化合物Ia中提取。B-Raf蛋白2可用于癌症研究[1]。

 B-Raf IN 2名称

英文名 B-Raf IN 2

 B-Raf IN 2生物活性

描述 B-Raf IN 2是一种有效的选择性BRAF抑制剂,从专利WO2021116055A1化合物Ia中提取。B-Raf蛋白2可用于癌症研究[1]。
相关类别
靶点

BRafV600E

体外研究 2中的B-Raf显示MAPK信号通路的旁氧激活显著减少,同时保持高效价[1]。
参考文献

[1]. Dolente C, et, al. New methylquinazolinone derivatives. WO2021116055A1.

 B-Raf IN 2物理化学性质

分子式 C20H17F2N5O4S
分子量 461.44
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