GRK6-IN-3

• 常用名: GRK6-IN-3
• 英文名: GRK6-IN-3
• CAS号: 499231-87-7
• 分子量: 312.37
• 密度: N/A
• 沸点: N/A
• 分子式: C₁₇H₂₀N₄O₂
• 熔点: N/A
• 闪点: N/A

GRK6-IN-3用途

GRK6-IN-3是一种G蛋白偶联受体6激酶(GRK6)抑制剂,其IC50为1.03μM[1]。

GRK6-IN-3名称

• 英文名: GRK6-IN-3

GRK6-IN-3生物活性

• 描述: GRK6-IN-3是一种G蛋白偶联受体6激酶(GRK6)抑制剂,其IC50为1.03μM[1]。
• 相关类别:
  研究领域 >> 炎症/免疫
• 靶点实验:

  IC50: 1.03 μM (GRK6)[1]

• 参考文献:

  [1]. Alexander Keith Stewart, et al. Inhibiting g protein coupled receptor 6 kinase polypeptides. WO2013063458A2.

GRK6-IN-3物理化学性质

• 分子式: C₁₇H₂₀N₄O₂
• 分子量: 312.37
• InChIKey: PEHCLEWOBIHBRW-UHFFFAOYSA-N
• SMILES: CCCCCn1c(N)c(C(=O)OC)c2nc3ccccc3nc21

GRK6-IN-3靶点实验

查看更多实验

实验名称：TBD from US Patent US10252984: "Inhibiting G protein coupled receptor 6 kinase polype... 来源：BindingDB 靶标：N/A External Id：BindingDB_2646_1

实验名称：Dicer-mediated maturation of pre-microRNA 来源：Center for Chemical Genomics, University of Michigan 靶标：N/A External Id：TargetID_659_CEMA

实验名称：Inhibitors of CDC25B-CDK2/CyclinA interaction 来源：Center for Chemical Genomics, University of Michigan External Id：MScreen:TargetID_600

实验名称：Cell-based high throughput primary assay to identify activators of GPR151 来源：The Scripps Research Institute Molecular Screening Center 靶标：RecName: Full=G-protein coupled receptor 151; AltName: Full=G-protein coupled receptor PGR7; AltName: Full=GPCR-2037; AltName: Full=Galanin receptor 4; AltName: Full=Galanin-receptor-like protein; Short=GalRL External Id：GPR151_PHUNTER_AG_LUMI_1536_1X%ACT

实验名称：AlphaScreen-based biochemical high throughput primary assay to identify activators of... 来源：The Scripps Research Institute Molecular Screening Center 靶标：N/A External Id：FBW7_ACT_ALPHA_1536_1X%ACT PRUN

实验名称：AlphaScreen-based biochemical high throughput primary assay to identify inhibitors of... 来源：The Scripps Research Institute Molecular Screening Center External Id：MITF_INH_Alpha_1536_1X%INH PRUN

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