Milveterol

• 常用名: Milveterol
• 英文名: Milveterol
• CAS号: 652990-07-3
• 分子量: 435.51500
• 密度: N/A
• 沸点: N/A
• 分子式: C₂₅H₂₉N₃O₄
• 熔点: N/A
• 闪点: N/A

Milveterol用途

Milveterol (GSK 159797) is a potent, selective long-acting β2 adrenoceptor agonist with pEC50 of 10.2 in cell-based assays, displays good β2/β1 selectivity (>300-fold).

Milveterol名称

• 英文名: N-[2-hydroxy-5-[(1R)-1-hydroxy-2-[2-[4-[[(2R)-2-hydroxy-2-phenylethyl]amino]phenyl]ethylamino]ethyl]phenyl]formamide

Milveterol物理化学性质

• 分子式: C₂₅H₂₉N₃O₄
• 分子量: 435.51500
• 精确质量: 435.21600
• PSA: 117.34000
• LogP: 4.08510
• InChIKey: BMKINZUHKYLSKI-DQEYMECFSA-N
• SMILES: O=CNc1cc(C(O)CNCCc2ccc(NCC(O)c3ccccc3)cc2)ccc1O

Milveterol靶点实验

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实验名称：Selectivity ratio of Ki for human beta1 adrenergic receptor to Ki for human beta2 adr... 来源：ChEMBL 靶标：N/A External Id：CHEMBL3369036

实验名称：Agonist activity at human beta1 adrenergic receptor expressed in cells by cAMP accumu... 来源：ChEMBL 靶标：Beta-1 adrenergic receptor External Id：CHEMBL3369037

实验名称：Displacement of [3H]dihydroalprenolol from human beta2 adrenergic receptor expressing... 来源：ChEMBL 靶标：Beta-2 adrenergic receptor External Id：CHEMBL3369035

实验名称：Agonist activity at recombinant human beta2-adrenoceptor expressed in whole cells ass... 来源：ChEMBL 靶标：Beta-2 adrenergic receptor External Id：CHEMBL1943768

实验名称：Agonist activity at human beta2 adrenergic receptor in human BEAS-2B cells by cAMP ac... 来源：ChEMBL 靶标：Beta-2 adrenergic receptor External Id：CHEMBL3369040

实验名称：Intrinsic activity at beta2-adrenoceptor endogenously expressed in human BEAS-2B cell... 来源：ChEMBL 靶标：Beta-2 adrenergic receptor External Id：CHEMBL1943771

实验名称：Displacement of [3H]dihydroalprenolol from beta2 receptor (unknown origin) by liquid ... 来源：ChEMBL 靶标：Beta-2 adrenergic receptor External Id：CHEMBL3294890

实验名称：Intrinsic agonist activity at human beta2 adrenergic receptor in human BEAS-2B cells ... 来源：ChEMBL 靶标：Beta-2 adrenergic receptor External Id：CHEMBL3369041

实验名称：Agonist activity at human recombinant beta2 receptor assessed as cAMP accumulation by... 来源：ChEMBL 靶标：Beta-2 adrenergic receptor External Id：CHEMBL3294889

实验名称：Agonist activity at human beta2 adrenergic receptor expressed in cells by cAMP accumu... 来源：ChEMBL 靶标：Beta-2 adrenergic receptor External Id：CHEMBL3369038

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Milveterol英文别名

• Milveterol
• UNII-LGY1VQ9622