Synthesis and stereochemical effects of pyrrolidinyl-acetylenic thieno [3, 2-d] pyrimidines as EGFR and ErbB-2 inhibitors

KL Stevens, KJ Alligood, JGB Alberti, TR Caferro…

Index: Bioorganic and Medicinal Chemistry Letters, , vol. 19, # 1 p. 21 - 26

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Citation Number: 13

Abstract

... Bioorganic & Medicinal Chemistry Letters. ... a Department of Oncology Medicinal Chemistry, GlaxoSmithKline, Research ... Biology, GlaxoSmithKline, Research Triangle Park, NC 27709, USA; c Department of Computational and Structural Chemistry, GlaxoSmithKline, Research ...