Tetrahedron

Synthesis of activated 3-substituted indoles: an optimised one-pot procedure

K Pchalek, AW Jones, MMT Wekking, DSC Black

Index: Pchalek, Karin; Jones, Ashley W.; Wekking, Monique M.T.; Black, David StC. Tetrahedron, 2005 , vol. 61, # 1 p. 77 - 82

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Citation Number: 42

Abstract

Download PDF Opens in a new window. Article suggestions will be shown in a dialog on return to ScienceDirect. ... Please enable JavaScript to use all the features on this page. ... 3-Substituted-4,6-dimethoxyindoles can be synthesised in a one-pot procedure from 3,5-dimethoxyaniline and 2-haloketones in the presence of lithium bromide and sodium bicarbonate. ... The indole nucleus is present in a wide range of natural products, and consequently a variety of ...