Enantioselective synthesis of Janus kinase inhibitor INCB018424 via an organocatalytic aza-Michael reaction

Q Lin, D Meloni, Y Pan, M Xia, J Rodgers…

Index: Organic Letters, , vol. 11, # 9 p. 1999 - 2002

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Citation Number: 117

Abstract

... Volume: Page: Digital Object Identifier (DOI). ... Organic Letters. ... Lett. , 2009, 11 (9), pp 1999–2002. DOI: 10.1021/ol900350k. Publication Date (Web): March 27, 2009. Copyright © 2009 American Chemical Society. ...