Modification of estrone at the 6, 16, and 17 positions: novel potent inhibitors of 17β-hydroxysteroid dehydrogenase type 1

GM Allan, HR Lawrence, J Cornet…

Index: Journal of Medicinal Chemistry, , vol. 49, # 4 p. 1325 - 1345

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Citation Number: 60

Abstract

... Journal of Medicinal Chemistry. ... Medicinal Chemistry, Department of Pharmacy and Pharmacology and Sterix Ltd., University of Bath, Claverton Down, BA2 7AY, UK, Endocrinology and Metabolic Medicine and Sterix Ltd., Faculty of Medicine, Imperial College London, St ...

A novel efficient approach to the Synthesis of 6??Oxo Ethiny...

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