Tetrahedron

First enantioselective synthesis of the novel antiinfective TAN-1057A via its aminomethyl-substituted dihydropyrimidinone heterocycle

VN Belov, M Brands, S Raddatz, J Krüger…

Index: Waki; Kitajima; Izumiya Synthesis, 1981 , vol. No.4, p. 266 - 268

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Citation Number: 12

Abstract

... An attempt to synthesize (S)-15 along a shorter route was made (Scheme 3). Curtius ... Diastereoselective synthesis of TAN-1057A ∗ 2HCl and its analogue with a β-lysine side chain: (a) hν ... 4b,d Therefore the pure diastereomer (3′S,5S)-21b was synthesized by coupling the ...