Tetrahedron Letters

Metal-free C–N bond-forming reaction: straightforward synthesis of anilines, through cleavage of aryl C–O bond and amide C–N bond

J Yu, P Zhang, J Wu, Z Shang

Index: Yu, Jianzhong; Zhang, Peizhi; Wu, Jun; Shang, Zhicai Tetrahedron Letters, 2013 , vol. 54, # 24 p. 3167 - 3170

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Citation Number: 5

Abstract

An efficient metal-free C–N bond forming reaction through cleavage of aryl C–O bond and amide C–N bond has been developed. This process represents a practical method for the facile construction of anilines with a broad substrate scope and wide functional group tolerance in moderate to excellent yields.

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