Organic Letters 2011-05-06

Copper-catalyzed trifluoromethylation of aryl and vinyl boronic acids with an electrophilic trifluoromethylating reagent.

Tianfei Liu, Qilong Shen

Index: Org. Lett. 13 , 2342-2345, (2011)

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Abstract

A copper-catalyzed trifluoromethylation of aryl- and alkenylboronic acids with Togni's reagent was described. The reaction proceeded in good to excellent yields for a range of different substrates including heteroarylboronic acids and substrates with a variety of functional groups under mild reaction conditions.

Structure	Name/CAS No.	Molecular Formula	Articles
	Togni's Reagent CAS:887144-97-0	C₁₀H₁₀F₃IO

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Copper-catalyzed trifluoromethylation of aryl and vinyl boronic acids with an electrophilic trifluoromethylating reagent.

Abstract

Related Compounds