Bioorganic & medicinal chemistry

Conformationally restrained carbazolone-containing α, γ-diketo acids as inhibitors of HIV integrase

X Li, R Vince

Index: Bioorganic and Medicinal Chemistry, , vol. 14, # 9 p. 2942 - 2955

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Citation Number: 53

Abstract

... Bioorganic & Medicinal Chemistry. ... Department of Medicinal Chemistry, College of ... 3). This modification afforded a 'drug-like' tricyclic carbazolone molecule, which is an important pharmacophore present in many pharmaceutical agents such as 5HT 3 inhibitors and anti-tumor ...

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