Name | PF-04577806 | CAS# | 1072100-81-2 | |
---|---|---|---|---|
Price | ¥Inquiry/100mg ¥Inquiry/250mg ¥Inquiry/1g | Purity | 98.0% | |
Stocking Period |
1 Day | Stock | 3 | |
Product Webpage: | https://www.dcchemicals.com/product_show-pf-04577806.html |
Detail
Product Information
PF-04577806 is a potent, selective and ATP competitive PKC inhibitor. PF-04577806 shows potent inhibitory activity towards PKCα, PKCβI, PKCβII, PKCγ, and PKCθ with IC50s of 2.4 nM, 8.1 nM, 6.9 nM, 45.9 nM, and 29.5 nM, respectively. PF-04577806 can reverse retinal vascular leakage in diabetic rats. |