Name | E3 ligase Ligand-Linker Conjugates 12 |
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Description | E3 ligase Ligand-Linker Conjugates 12 is a synthesized compound that incorporates an E3 ligase ligand and a linker used in PROTAC technology. |
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Related Catalog | |
Target |
E3 Ligase Ligand-Linker Conjugate[1] |
In Vitro | E3 ligase Ligand-Linker Conjugates 12 is extracted from patent WO/2016/146985A1, figure 11. PROTAC has been developed having structure A-L-B that can tether a bromodomain inhibitor via a moiety which binds to a protein within the bromo- and Extra-terminal (BET) family of proteins to a small molecule E3 ubiquintin ligase protein binding ligand compond via a suitable linker[1][2]. |
References |
[1]. WO/2016/146985A1 |
Molecular Formula | C30H43N7O7S |
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Molecular Weight | 645.77 |