DC Chemicals Limited
China
Product Name: BAY-1316957
Price: $Inquiry/100mg $Inquiry/250mg $Inquiry/1g
Purity: 98.0%
Stocking Period: 3 Day
Contact: Tony Cao

1613264-40-6

1613264-40-6 structure

1613264-40-6 structure

Name: BAY-1316957
Chemical Name: BAY-1316957
CAS Number: 1613264-40-6
Molecular Formula: C₂₇H₂₇N₃O₃
Molecular Weight: 441.52
Catalog: Signaling Pathways GPCR/G Protein Prostaglandin Receptor
Create Date: 2019-03-31 01:09:34
Modify Date: 2024-01-27 16:26:28
BAY-1316957 is a highly potent and selective EP4 receptor antagonist with an IC50 of 15.3 nM. Good oral bioavailability[1].

Name	BAY-1316957

Description	BAY-1316957 is a highly potent and selective EP4 receptor antagonist with an IC50 of 15.3 nM. Good oral bioavailability[1].
Related Catalog	Signaling Pathways >> GPCR/G Protein >> Prostaglandin Receptor Research Areas >> Inflammation/Immunology
Target	IC50: 15.3 nM (EP4)[1]
References	[1]. Bäurle S, et al. Identification of a Benzimidazolecarboxylic Acid Derivative (BAY 1316957) as a Potent and Selective Human Prostaglandin E2 Receptor Subtype 4 (hEP4-R) Antagonist for the Treatment of Endometriosis. J Med Chem. 2019 Mar 14;62(5):2541-2563.

Molecular Formula	C₂₇H₂₇N₃O₃
Molecular Weight	441.52