939391-31-8

939391-31-8 structure

Name: CETP-IN-3
Chemical Name: CETP-IN-3
CAS Number: 939391-31-8
Molecular Formula: C₃₀H₂₄F₁₂N₂O₄
Molecular Weight: 704.50
Catalog: Signaling Pathways Metabolic Enzyme/Protease CETP
Create Date: 2019-08-03 19:47:59
Modify Date: 2024-01-09 15:51:24
CETP-IN-3 (Compound 13) is an small molecule inhibitor of the plasma glycoprotein cholesterol ester transfer protein (CETP), elevating HDL-C through inhibition of CETP. CETP-IN-3 for the CETP inhibitory activity in the scintillation proximity (SPA) and whole plasma assay (WPA) with IC50s of 0.002 μM and 0.06 μM, respectively[1].

Name	CETP-IN-3

Description	CETP-IN-3 (Compound 13) is an small molecule inhibitor of the plasma glycoprotein cholesterol ester transfer protein (CETP), elevating HDL-C through inhibition of CETP. CETP-IN-3 for the CETP inhibitory activity in the scintillation proximity (SPA) and whole plasma assay (WPA) with IC50s of 0.002 μM and 0.06 μM, respectively[1].
Related Catalog	Research Areas >> Cardiovascular Disease Signaling Pathways >> Metabolic Enzyme/Protease >> CETP
References	[1]. Finlay HJ, et al. Discovery of a Lead Triphenylethanamine Cholesterol Ester Transfer Protein (CETP) Inhibitor. ACS Med Chem Lett. 2019 May 6; 10(6):911-916.

Molecular Formula	C₃₀H₂₄F₁₂N₂O₄
Molecular Weight	704.50