Name | ACG-548B |
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Description | A potent, selective choline kinase α (ChoKα) inhibitor with IC50 of 0.12 uM, >400-fold selectivity over ChoKβ; demonstrates in vitro antiproliferative activity against HT29 cells with IC50 of 2.08 uM. |
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References | References 1. Lacal JC, et al. Mol Cancer Ther. 2015 Jan;14(1):31-9. 2. Patent US 20110178124 A1. Pyridinium and quinolinium derivatives. View Related Products by Target Choline Kinase (ChoK) |
Molecular Formula | C38H34Br2Cl2N4 |
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Molecular Weight | 777.426 |