442150-41-6
442150-41-6 structure
- Name: CSV0C018875
- Chemical Name: CSV0C018875
- CAS Number: 442150-41-6
- Molecular Formula: C18H17ClN2O
- Molecular Weight: 312.79
- Catalog: Signaling Pathways Epigenetics Histone Methyltransferase
- Create Date: 2021-09-13 00:34:30
- Modify Date: 2024-01-09 17:35:38
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CSV0C018875 is a quinoline-based EHMT2/G9a inhibitor. CSV0C018875 exhibits lesser cytotoxicity than BIX-01294[1].
| Name | CSV0C018875 |
|---|
| Description | CSV0C018875 is a quinoline-based EHMT2/G9a inhibitor. CSV0C018875 exhibits lesser cytotoxicity than BIX-01294[1]. |
|---|---|
| Related Catalog | |
| Target |
G9a |
| In Vitro | CSV0C018875 (2.5-20 μM; 48 hours) inhibits the levels of H3K9me2 modifications in the histones[1]. Western Blot Analysis[1] Cell Line: HEK293 cells Concentration: 2.5 μM, 10 μM, 20 μM Incubation Time: 48 hours Result: Inhibited the enzymatic activity of G9a in a dose-dependent manner in HEK293 cells. |
| References |
| Molecular Formula | C18H17ClN2O |
|---|---|
| Molecular Weight | 312.79 |