2215931-60-3
2215931-60-3 structure
- Name: PCSK9 degrader 1
- Chemical Name: PCSK9 degrader 1
- CAS Number: 2215931-60-3
- Molecular Formula: C34H34FN3O6S
- Molecular Weight: 631.71
- Catalog: Signaling Pathways Metabolic Enzyme/Protease Ser/Thr Protease
- Create Date: 2021-10-07 19:47:50
- Modify Date: 2024-01-10 12:25:03
-
PCSK9 degrader 1 is a selective proprotein convertase substilisin-like/kexin type 9 (PCSK9) degrader. PCSK9 degrader 1 does not affect PCSK9 function[1].
| Name | PCSK9 degrader 1 |
|---|
| Description | PCSK9 degrader 1 is a selective proprotein convertase substilisin-like/kexin type 9 (PCSK9) degrader. PCSK9 degrader 1 does not affect PCSK9 function[1]. |
|---|---|
| Related Catalog | |
| In Vitro | Biphenyl acid PCSK9 degrader 1 (compound 9) binds to and thermally stabilizes PCSK9 in a complex environment such as Huh7 lysate[1]. PCSK9 degrader 1 (compound 9), with high affinity for recombinant PCSK9 and target engagement in cell lysate, could be used as a recruiting element to promote the selective degradation of PCSK9[1]. |
| References |
| Molecular Formula | C34H34FN3O6S |
|---|---|
| Molecular Weight | 631.71 |