2630904-45-7
2630904-45-7 structure
- Name: MRTX-1719
- Chemical Name: MRTX-1719
- CAS Number: 2630904-45-7
- Molecular Formula: C23H18ClFN6O2
- Molecular Weight: 464.88
- Catalog: Signaling Pathways Epigenetics Histone Methyltransferase
- Create Date: 2021-12-27 08:44:34
- Modify Date: 2024-01-08 20:21:35
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MRTX-1719 is a potent first-in-class selective inhibitor of the PRMT5/MTA complex, with an IC50 of less than 10 nM in PRMT5/MTA MTAPDEL SDMA cells[1].
| Name | MRTX-1719 |
|---|
| Description | MRTX-1719 is a potent first-in-class selective inhibitor of the PRMT5/MTA complex, with an IC50 of less than 10 nM in PRMT5/MTA MTAPDEL SDMA cells[1]. |
|---|---|
| Related Catalog | |
| Target |
IC50: <10 nM (PRMT5/MTA MTAPDEL SDMA cells)[1]. |
| References |
[1]. Targeting the genetic and immunological drivers of cancer. |
| Molecular Formula | C23H18ClFN6O2 |
|---|---|
| Molecular Weight | 464.88 |