Shanghai Nianxing Industrial Co., Ltd
China
Product Name: CCG-271423
Price: Check
Purity: 98.0%
Stocking Period: 10 Day
Contact: Yang
Email: sales@echemcloud.com

DC Chemicals Limited
China
Product Name: CCG-271423
Price: ￥Inquiry/100mg ￥Inquiry/250mg ￥Inquiry/1g
Purity: 98.0%
Stocking Period: 10 Day
Contact: Tony Cao
Email: sales@dcchemicals.com

2750413-88-6

2750413-88-6 structure

2750413-88-6 structure

Name: CCG-271423
Chemical Name: CCG-271423
CAS Number: 2750413-88-6
Molecular Formula: C₂₈H₂₆N₄O₃
Molecular Weight: 466.53
Catalog: Research Areas Cardiovascular Disease
Create Date: 2022-09-10 09:07:10
Modify Date: 2025-08-26 23:30:38
CCG-271423 is a potent and selective GRK5 inhibitor with IC50 values of 0.0021 μM and 44 μM for GRK5 and GRK2, respectively. CCG-271423 inhibits cardiomyocyte contractility and decreases in Ca2+ transience[1].

Name	CCG-271423

Description	CCG-271423 is a potent and selective GRK5 inhibitor with IC50 values of 0.0021 μM and 44 μM for GRK5 and GRK2, respectively. CCG-271423 inhibits cardiomyocyte contractility and decreases in Ca2+ transience[1].
Related Catalog	Research Areas >> Cardiovascular Disease
Target	IC50: 0.0021 μM (GRK5) and 44 μM (GRK5)[1]
In Vitro	CCG-271423 (1 μM) does not alter cardiomyocyte contractility and decreases in Ca2+ transience[1].
References	[1]. Rowlands R, et, al. Expanding the Arsenal: Development of G-Protein Receptor Kinase 5 Inhibitors Utilizing a Covalent Strategy.

Molecular Formula	C₂₈H₂₆N₄O₃
Molecular Weight	466.53

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