2750413-88-6
2750413-88-6 structure
- Name: CCG-271423
- Chemical Name: CCG-271423
- CAS Number: 2750413-88-6
- Molecular Formula: C28H26N4O3
- Molecular Weight: 466.53
- Catalog: Research Areas Cardiovascular Disease
- Create Date: 2022-09-10 09:07:10
- Modify Date: 2024-04-07 11:49:46
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CCG-271423 is a potent and selective GRK5 inhibitor with IC50 values of 0.0021 μM and 44 μM for GRK5 and GRK2, respectively. CCG-271423 inhibits cardiomyocyte contractility and decreases in Ca2+ transience[1].
| Name | CCG-271423 |
|---|
| Description | CCG-271423 is a potent and selective GRK5 inhibitor with IC50 values of 0.0021 μM and 44 μM for GRK5 and GRK2, respectively. CCG-271423 inhibits cardiomyocyte contractility and decreases in Ca2+ transience[1]. |
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| Related Catalog | |
| Target |
IC50: 0.0021 μM (GRK5) and 44 μM (GRK5)[1] |
| In Vitro | CCG-271423 (1 μM) does not alter cardiomyocyte contractility and decreases in Ca2+ transience[1]. |
| References |
| Molecular Formula | C28H26N4O3 |
|---|---|
| Molecular Weight | 466.53 |