CCG-271423
Modify Date: 2024-04-07 11:49:46
CCG-271423 structure
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Common Name | CCG-271423 | ||
|---|---|---|---|---|
| CAS Number | 2750413-88-6 | Molecular Weight | 466.53 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C28H26N4O3 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of CCG-271423CCG-271423 is a potent and selective GRK5 inhibitor with IC50 values of 0.0021 μM and 44 μM for GRK5 and GRK2, respectively. CCG-271423 inhibits cardiomyocyte contractility and decreases in Ca2+ transience[1]. |
| Name | CCG-271423 |
|---|
| Description | CCG-271423 is a potent and selective GRK5 inhibitor with IC50 values of 0.0021 μM and 44 μM for GRK5 and GRK2, respectively. CCG-271423 inhibits cardiomyocyte contractility and decreases in Ca2+ transience[1]. |
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| Related Catalog | |
| Target |
IC50: 0.0021 μM (GRK5) and 44 μM (GRK5)[1] |
| In Vitro | CCG-271423 (1 μM) does not alter cardiomyocyte contractility and decreases in Ca2+ transience[1]. |
| References |
| Molecular Formula | C28H26N4O3 |
|---|---|
| Molecular Weight | 466.53 |