1152810-23-5

1152810-23-5 structure

Name: Sheng Gelieting
Chemical Name: Sheng Gelieting
CAS Number: 1152810-23-5
Molecular Formula: C₁₇H₁₆F₆N₄O
Molecular Weight: 406.33
Catalog: Signaling Pathways Metabolic Enzyme/Protease Dipeptidyl Peptidase
Create Date: 2022-11-21 11:27:02
Modify Date: 2025-08-21 20:14:14
Sheng Gelieting (CGT-8012) is a dipeptidy peptidase-IV enzyme (DP-IV) inhibitor. Sheng Gelieting has great DP-IV inhibition activity with an IC50 value of 87 nM. Sheng Gelieting can be used for curing or preventing diseases relevant to the dipeptidy peptidase-IV enzyme, such as the diabetes, particularly the II-type diabete[1].

Name	Sheng Gelieting

Description	Sheng Gelieting (CGT-8012) is a dipeptidy peptidase-IV enzyme (DP-IV) inhibitor. Sheng Gelieting has great DP-IV inhibition activity with an IC50 value of 87 nM. Sheng Gelieting can be used for curing or preventing diseases relevant to the dipeptidy peptidase-IV enzyme, such as the diabetes, particularly the II-type diabete[1].
Related Catalog	Research Areas >> Endocrinology Signaling Pathways >> Metabolic Enzyme/Protease >> Dipeptidyl Peptidase
Target	IC50: 87 nM (DP-IV)[1]
In Vitro	Sheng Gelieting has great dipeptidy peptidase-IV enzyme (DP-IV) inhibition activity with an IC50 value of 87 nM[1].
References	[1]. Qiang Yu, et al. Beta-amino tetrahydropyrazine, tetrahydropyrimidine and tetrahydropyridine used as dipeptidy peptidase inhibitors for curing or preventing diabetes. Patent. CN101899047A.

Molecular Formula	C₁₇H₁₆F₆N₄O
Molecular Weight	406.33