Name | Blue FPG-A trisodium |
---|
Description | Blue FPG-A trisodium is a selective antagonist of P2X1 receptor and P2Y1 receptor with IC50 values of 35.5 μM and 2.6 μM, respectively. Blue FPG-A trisodium is a structural isomer of the components of Reactive Blue 2 (RB2)[1]. |
---|---|
Related Catalog | |
Target |
p2x1 Receptor:35.5 μM (IC50) P2Y1 Receptor:2.6 μM (IC50) |
In Vitro | Blue FPG-A trisodium (RB 2 para) (1、3.2、10、32 和 100 μM) 抑制 α、β-亚甲基 ATP (α、β-MeATP) 诱导的大鼠输精管 (RVD) 收缩和 5’-o-(2-硫代二磷酸腺苷) (ADPβS) 诱导的卡巴胆碱 (Carbachol,HY-B1208) 预处理的豚鼠大肠带绦虫 (GPTC) 的松弛[1]。 |
References |
Molecular Formula | C29H17ClN7Na3O11S3 |
---|---|
Molecular Weight | 840.10 |