| Name | Cbl-b-IN-7 |
|---|
| Description | Cbl-b-IN-7 (Compound 248) is a casitas B-lineage lymphoma-b (Cbl-b) and c-Cbl inhibitor with IC50s of 6.7 nM and 5.2 nM, respectively[1]. |
|---|---|
| Related Catalog | |
| Target |
IC50: 5.2 nM (c-Cbl), 6.7 nM (Cbl-b)[1] |
| References |
[1]. Jun Liang, et al. Lactams as cbl-b inhibitors. Patent WO2022169997A1. |
| Molecular Formula | C29H31F4N5O2 |
|---|---|
| Molecular Weight | 557.58 |