217438-17-0
217438-17-0 structure
- Name: SB 268262
- Chemical Name: N-Methyl-N-(2-methylphenyl)-3-nitro-4-(1,3-thiazol-2-ylsulfinyl)b enzamide
- CAS Number: 217438-17-0
- Molecular Formula: C18H15N3O4S2
- Molecular Weight: 401.46
- Catalog: Research Areas Neurological Disease
- Create Date: 2018-10-23 15:04:59
- Modify Date: 2025-08-27 00:44:18
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CGRP antagonist 4 is an antagonist of calcitonin gene-related peptide (CGRP) receptor. CGRP antagonist 4 shows the highest affinity for CGRP receptors in the human brain. CGRP antagonist 4 can be used to study the binding properties of non-peptide calcitonin gene-related peptide (CGRP) receptor antagonist (gepants) in rat, pig and human menes [1].
| Name | N-Methyl-N-(2-methylphenyl)-3-nitro-4-(1,3-thiazol-2-ylsulfinyl)b enzamide |
|---|---|
| Synonyms | (+/-)-SB-273779 N-Methyl-N-(2-methylphenyl)-3-nitro-4-(2-thiazolylsulfinyl)-benzamide |
| Description | CGRP antagonist 4 is an antagonist of calcitonin gene-related peptide (CGRP) receptor. CGRP antagonist 4 shows the highest affinity for CGRP receptors in the human brain. CGRP antagonist 4 can be used to study the binding properties of non-peptide calcitonin gene-related peptide (CGRP) receptor antagonist (gepants) in rat, pig and human menes [1]. |
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| Related Catalog | |
| References |
| Molecular Formula | C18H15N3O4S2 |
|---|---|
| Molecular Weight | 401.46 |
| Exact Mass | 401.05000 |
| PSA | 143.54000 |
| LogP | 5.19190 |
| Symbol |
GHS07 |
|---|---|
| Signal Word | Warning |
| Hazard Statements | H302-H319 |
| Precautionary Statements | P305 + P351 + P338 |
| RIDADR | NONH for all modes of transport |