Name | Somatostatin Antagonist |
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Synonyms |
Cyclosomatostatin
C[AMINOHEPTANOYL-PHE-DTRP-LYS-THR: BZL] 6-(4-aminobutyl)-12-benzyl-9-(1H-indol-3-ylmethyl)-3-(1-phenylmethoxyethyl)-1,4,7,10,13-pentazacycloicosane-2,5,8,11,14-pentone Cyclo(7-Aminoheptanoyl-Phe-D-Trp-Lys-Thr[Bzl]) |
Description | Cyclosomatostatin is a potent somatostatin (SST) receptor antagonist. Cyclosomatostatin can inhibit somatostatin receptor type 1 (SSTR1) signaling and decreases cell proliferation, ALDH+ cell population size and sphere-formation in colorectal cancer (CRC) cells[1]. |
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Related Catalog | |
References |
Density | 1.147g/cm3 |
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Boiling Point | 1118.4ºC at 760 mmHg |
Molecular Formula | C44H57N7O6 |
Molecular Weight | 779.96700 |
Flash Point | 630.2ºC |
Exact Mass | 779.43700 |
PSA | 196.54000 |
LogP | 6.05120 |
Index of Refraction | 1.558 |
Storage condition | -20°C |
Personal Protective Equipment | Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter |
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RIDADR | NONH for all modes of transport |
WGK Germany | 3 |