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84211-54-1

84211-54-1 structure
84211-54-1 structure
  • Name: Cyclosomatostatin
  • Chemical Name: Somatostatin Antagonist
  • CAS Number: 84211-54-1
  • Molecular Formula: C44H57N7O6
  • Molecular Weight: 779.96700
  • Catalog: Signaling Pathways GPCR/G Protein Somatostatin Receptor
  • Create Date: 2017-05-15 17:41:29
  • Modify Date: 2024-01-02 15:12:07
  • Cyclosomatostatin is a potent somatostatin (SST) receptor antagonist. Cyclosomatostatin can inhibit somatostatin receptor type 1 (SSTR1) signaling and decreases cell proliferation, ALDH+ cell population size and sphere-formation in colorectal cancer (CRC) cells[1].

Name Somatostatin Antagonist
Synonyms Cyclosomatostatin
C[AMINOHEPTANOYL-PHE-DTRP-LYS-THR: BZL]
6-(4-aminobutyl)-12-benzyl-9-(1H-indol-3-ylmethyl)-3-(1-phenylmethoxyethyl)-1,4,7,10,13-pentazacycloicosane-2,5,8,11,14-pentone
Cyclo(7-Aminoheptanoyl-Phe-D-Trp-Lys-Thr[Bzl])
Description Cyclosomatostatin is a potent somatostatin (SST) receptor antagonist. Cyclosomatostatin can inhibit somatostatin receptor type 1 (SSTR1) signaling and decreases cell proliferation, ALDH+ cell population size and sphere-formation in colorectal cancer (CRC) cells[1].
Related Catalog
References

[1]. Shirin R Modarai, et al. Somatostatin signaling via SSTR1 contributes to the quiescence of colon cancer stem cells. BMC Cancer. 2016 Dec 7;16(1):941.

Density 1.147g/cm3
Boiling Point 1118.4ºC at 760 mmHg
Molecular Formula C44H57N7O6
Molecular Weight 779.96700
Flash Point 630.2ºC
Exact Mass 779.43700
PSA 196.54000
LogP 6.05120
Index of Refraction 1.558
Storage condition -20°C
Personal Protective Equipment Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter
RIDADR NONH for all modes of transport
WGK Germany 3