Cyclosomatostatin

Modify Date: 2024-01-02 15:12:07

Cyclosomatostatin structure	Common Name	Cyclosomatostatin
	CAS Number	84211-54-1	Molecular Weight	779.96700
	Density	1.147g/cm3	Boiling Point	1118.4ºC at 760 mmHg
	Molecular Formula	C₄₄H₅₇N₇O₆	Melting Point	N/A
	MSDS	USA	Flash Point	630.2ºC

Use of Cyclosomatostatin

Cyclosomatostatin is a potent somatostatin (SST) receptor antagonist. Cyclosomatostatin can inhibit somatostatin receptor type 1 (SSTR1) signaling and decreases cell proliferation, ALDH+ cell population size and sphere-formation in colorectal cancer (CRC) cells[1].

Name	Somatostatin Antagonist
Synonym	More Synonyms

Description	Cyclosomatostatin is a potent somatostatin (SST) receptor antagonist. Cyclosomatostatin can inhibit somatostatin receptor type 1 (SSTR1) signaling and decreases cell proliferation, ALDH+ cell population size and sphere-formation in colorectal cancer (CRC) cells[1].
Related Catalog	Research Areas >> Cancer Signaling Pathways >> GPCR/G Protein >> Somatostatin Receptor
References	[1]. Shirin R Modarai, et al. Somatostatin signaling via SSTR1 contributes to the quiescence of colon cancer stem cells. BMC Cancer. 2016 Dec 7;16(1):941.

Density	1.147g/cm3
Boiling Point	1118.4ºC at 760 mmHg
Molecular Formula	C₄₄H₅₇N₇O₆
Molecular Weight	779.96700
Flash Point	630.2ºC
Exact Mass	779.43700
PSA	196.54000
LogP	6.05120
Index of Refraction	1.558
Storage condition	-20°C

Cyclosomatostatin MSDS(Chinese)

Personal Protective Equipment	Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter
RIDADR	NONH for all modes of transport
WGK Germany	3

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Cyclosomatostatin

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