1044535-52-5

1044535-52-5 structure

Name: Dagrocorat
Chemical Name: (4bS,7R,8aR)-4b-benzyl-7-hydroxy-N-(2-methylpyridin-3-yl)-7-(trifluoromethyl)-5,6,8,8a,9,10-hexahydrophenanthrene-2-carboxamide
CAS Number: 1044535-52-5
Molecular Formula: C₂₉H₂₉F₃N₂O₂
Molecular Weight: 494.54800
Catalog: Signaling Pathways GPCR/G Protein Glucocorticoid Receptor
Create Date: 2016-11-19 19:20:41
Modify Date: 2025-08-26 21:25:54
Dagrocorat (PF-00251802) is a novel and dissociated glucocorticoid receptor agonist.

Name	(4bS,7R,8aR)-4b-benzyl-7-hydroxy-N-(2-methylpyridin-3-yl)-7-(trifluoromethyl)-5,6,8,8a,9,10-hexahydrophenanthrene-2-carboxamide
Synonyms	unii-opm23un90u

Description	Dagrocorat (PF-00251802) is a novel and dissociated glucocorticoid receptor agonist.
Related Catalog	Signaling Pathways >> GPCR/G Protein >> Glucocorticoid Receptor Research Areas >> Inflammation/Immunology
References	[1]. Ripp SL,et al. In Vitro and In Vivo Investigation of Potential for Complex CYP3A Interaction for PF-00251802 (Dagrocorat), a Novel Dissociated Agonist of the Glucocorticoid Receptor. Clin Pharmacol Drug Dev. 2018 Mar;7(3):244-255.