85286-38-0
85286-38-0 structure
- Name: (D-Thr2)-Leu-Enkephalin-Thr
- Chemical Name: [D-Thr2,Leu5]enkephalin-Thr
- CAS Number: 85286-38-0
- Molecular Formula: C34H48N6O10
- Molecular Weight: 700.779
- Catalog: Signaling Pathways GPCR/G Protein Opioid Receptor
- Create Date: 2016-07-28 14:42:25
- Modify Date: 2024-01-09 20:11:34
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Deltakephalin is a potent, selective opiate δ-receptor agonist. Deltakephalin has analgesic properties[1].
| Name | [D-Thr2,Leu5]enkephalin-Thr |
|---|---|
| Synonyms |
D-Allothreonine, L-tyrosyl-D-threonylglycyl-L-phenylalanyl-L-leucyl-
(D-Thr2)-Leu-Enkephalin-Thr (D-Thr2)-Leu-Enkephalin-Thr, DTLET, Deltakephalin Tyr-D-Thr-Gly-Phe-Leu-Thr L-Tyrosyl-D-threonylglycyl-L-phenylalanyl-L-leucyl-D-allothreonine |
| Description | Deltakephalin is a potent, selective opiate δ-receptor agonist. Deltakephalin has analgesic properties[1]. |
|---|---|
| Related Catalog | |
| In Vivo | Deltakephalin (2 nM/rat; ICV; once) produces a pronounced analgesia in rats[1]. Animal Model: Male spontaneously hypertensive rats (SHR/n/Ibm) and male Wistar Albino Glaxo rats (WAG) (250-300 g)[1] Dosage: 2 nM/rat Administration: Intracerebroventrical injection Result: Produced pronounced analgesia in male spontaneously hypertensive rats with EC50 values of 0.57 and 0.88 nM for the tail flick test and the tail compression test, respectively. |
| Density | 1.3±0.1 g/cm3 |
|---|---|
| Boiling Point | 1155.4±65.0 °C at 760 mmHg |
| Molecular Formula | C34H48N6O10 |
| Molecular Weight | 700.779 |
| Flash Point | 652.5±34.3 °C |
| Exact Mass | 700.343201 |
| PSA | 269.51000 |
| LogP | 1.44 |
| Vapour Pressure | 0.0±0.3 mmHg at 25°C |
| Index of Refraction | 1.588 |