H4R antagonist 3

Modify Date: 2024-04-10 15:52:01

H4R antagonist 3 Structure
H4R antagonist 3 structure
Common Name H4R antagonist 3
CAS Number 1003091-20-0 Molecular Weight 372.91
Density N/A Boiling Point N/A
Molecular Formula C19H21ClN4S Melting Point N/A
MSDS N/A Flash Point N/A

 Use of H4R antagonist 3


H4R antagonist 3 (Example 18) is a histamine-4 receptor antagonist with an EC50 of <10 mM. H4R antagonist 3 can be used for the research of prevention of inflammatory, autoimmune, allergic, and ocular diseases[1].

 Names

Name WAY-621360-A
Synonym More Synonyms

 H4R antagonist 3 Biological Activity

Description H4R antagonist 3 (Example 18) is a histamine-4 receptor antagonist with an EC50 of <10 mM. H4R antagonist 3 can be used for the research of prevention of inflammatory, autoimmune, allergic, and ocular diseases[1].
Related Catalog
Target

EC50: <10 mM (histamine-4 receptor)[1]

References

[1]. Allen J. Borchardt, et al. Aminopyrimidine inhibitors of histamine receptors for the treatment of disease. Patent US20100063047A1.

 Chemical & Physical Properties

Molecular Formula C19H21ClN4S
Molecular Weight 372.91

 Synonyms

Thieno[2,3-d]pyrimidin-4-amine, 5-(4-chlorophenyl)-N-methyl-N-(1-methyl-4-piperidinyl)-