MK-3901
Modify Date: 2023-05-27 10:46:43
MK-3901 structure
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Common Name | MK-3901 | ||
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| CAS Number | 1149750-69-5 | Molecular Weight | 481.531 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C28H24FN5O2 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of MK-3901MK-3901 is a potent, selective, orally active P2X3 antagonist with IC50 of 21 nM; demonstrates efficacy similar to that of naproxen, after 60 mg/kg (p.o.) administration with EC90 of approximately 3 uM in the rat CFA model of inflammatory pain. |
| Name | MK-3901 |
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| Description | MK-3901 is a potent, selective, orally active P2X3 antagonist with IC50 of 21 nM; demonstrates efficacy similar to that of naproxen, after 60 mg/kg (p.o.) administration with EC90 of approximately 3 uM in the rat CFA model of inflammatory pain. |
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| References | References 1. Ginnetti AT, et al. Bioorg Med Chem Lett. 2018 May 1;28(8):1392-1396. View Related Products by Target P2X Receptor |
| Molecular Formula | C28H24FN5O2 |
|---|---|
| Molecular Weight | 481.531 |