Carbamazepine 10,11-epoxide-13C,d2

Modify Date: 2024-01-04 20:37:39

Carbamazepine 10,11-epoxide-13C,d2 Structure
Carbamazepine 10,11-epoxide-13C,d2 structure
Common Name Carbamazepine 10,11-epoxide-13C,d2
CAS Number 1189497-48-0 Molecular Weight 255.27
Density N/A Boiling Point N/A
Molecular Formula C1413CH10D2N2O2 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Carbamazepine 10,11-epoxide-13C,d2


Carbamazepine 10,11-epoxide-13C,d2 is the deuterium labeled Carbamazepine 10,11-epoxide-C13. Carbamazepine 10,11-epoxide-C13 is a 13C-labled Carbamazepine 10,11-epoxide. Carbamazepine 10,11-epoxide is an orally active metabolite of Carbamazepine (HY-B0246). Carbamazepine has anticonvulsant effect. Carbamazepine can be used for the research of seizures[1][2].

 Names

Name Carbamazepine 10,11-epoxide-13C,d2

 Carbamazepine 10,11-epoxide-13C,d2 Biological Activity

Description Carbamazepine 10,11-epoxide-13C,d2 is the deuterium labeled Carbamazepine 10,11-epoxide-C13. Carbamazepine 10,11-epoxide-C13 is a 13C-labled Carbamazepine 10,11-epoxide. Carbamazepine 10,11-epoxide is an orally active metabolite of Carbamazepine (HY-B0246). Carbamazepine has anticonvulsant effect. Carbamazepine can be used for the research of seizures[1][2].
Related Catalog
In Vitro Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].
References

[1]. Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019 Feb;53(2):211-216.  

[2]. T Tomson, et al. Single-dose kinetics and metabolism of carbamazepine-10,11-epoxide. Clin Pharmacol Ther. 1983 Jan;33(1):58-65.  

 Chemical & Physical Properties

Molecular Formula C1413CH10D2N2O2
Molecular Weight 255.27