(±)-Anatoxin A fumarate
Modify Date: 2024-01-07 17:19:30
(±)-Anatoxin A fumarate structure
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Common Name | (±)-Anatoxin A fumarate | ||
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| CAS Number | 1219922-30-1 | Molecular Weight | 281.304 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C14H19NO5 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of (±)-Anatoxin A fumarate(±)-Anatoxin A fumarate is a natural alkaloid isolated from freshwater cyanobacterium.(±)-Anatoxin A fumarate is a potent nicotinic receptor agonist and exhibits Ki values of 1.25 nM and 1.84 μM for binding to putative α4β2-type nAChR and α7-type nAChR in rat brain membranes, respectively. (±)-Anatoxin A fumarate stimulates [3H]-dopamine release from rat striatal synaptosomes (EC50=134 nM)[1]. |
| Name | 1-(9-Azabicyclo[4.2.1]non-2-en-2-yl)ethanone (2E)-2-butenedioate (1:1) |
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| Synonym | More Synonyms |
| Description | (±)-Anatoxin A fumarate is a natural alkaloid isolated from freshwater cyanobacterium.(±)-Anatoxin A fumarate is a potent nicotinic receptor agonist and exhibits Ki values of 1.25 nM and 1.84 μM for binding to putative α4β2-type nAChR and α7-type nAChR in rat brain membranes, respectively. (±)-Anatoxin A fumarate stimulates [3H]-dopamine release from rat striatal synaptosomes (EC50=134 nM)[1]. |
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| Related Catalog | |
| Target |
Ki: 1.25 nM ( α4β2 receptor) Ki: 1.84 μM ( α7 receptor)[1] |
| References |
| Molecular Formula | C14H19NO5 |
|---|---|
| Molecular Weight | 281.304 |
| Exact Mass | 281.126312 |
| PSA | 103.70000 |
| LogP | 1.45680 |
| Ethanone, 1-(9-azabicyclo[4.2.1]non-2-en-2-yl)-, (2E)-2-butenedioate (1:1) |
| 1-(9-Azabicyclo[4.2.1]non-2-en-2-yl)ethanone (2E)-2-butenedioate (1:1) |