![]() XD14 structure
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Common Name | XD14 | ||
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CAS Number | 1370888-71-3 | Molecular Weight | 421.510 | |
Density | 1.3±0.1 g/cm3 | Boiling Point | N/A | |
Molecular Formula | C20H27N3O5S | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of XD14XD14 is a BET bromodomain inhibitor with Kd values of 160, 170, 380, 490, 830 and 850 nM for BRD4(1), BRD2(1), BRD3(1), BRD3(2), BRD2(2) and BRD4(2) respectively. |
Name | XD14 |
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Synonym | More Synonyms |
Description | XD14 is a BET bromodomain inhibitor with Kd values of 160, 170, 380, 490, 830 and 850 nM for BRD4(1), BRD2(1), BRD3(1), BRD3(2), BRD2(2) and BRD4(2) respectively. |
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In Vitro | BET bromodomain inhibitor with Kd values of 160, 170, 380, 490, 830 and 850 nM for BRD4(1), BRD2(1), BRD3(1), BRD3(2), BRD2(2) and BRD4(2) respectively. XD14 also inhibits BRDT(1), CBP, p300 and BRDT(2) with Kd values of 1.2, 1.6, 2.6 and 3.7 ��M respectively. |
Density | 1.3±0.1 g/cm3 |
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Molecular Formula | C20H27N3O5S |
Molecular Weight | 421.510 |
Exact Mass | 421.167145 |
LogP | 2.38 |
Index of Refraction | 1.592 |
Storage condition | -20°C |
1H-Pyrrole-2-carboxamide, 4-acetyl-N-[5-[(diethylamino)sulfonyl]-2-hydroxyphenyl]-3-ethyl-5-methyl- |
XD14 |
4-Acetyl-N-[5-(diethylsulfamoyl)-2-hydroxyphenyl]-3-ethyl-5-methyl-1H-pyrrole-2-carboxamide |
MFCD23144071 |