KT203
Modify Date: 2024-01-04 13:31:09
KT203 structure
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Common Name | KT203 | ||
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| CAS Number | 1402612-64-9 | Molecular Weight | 466.53 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C28H26N4O3 | Melting Point | N/A | |
| MSDS | USA | Flash Point | N/A | |
Use of KT203KT203 is a potent and selective inhibitor of α/β-hydrolase domain containing 6 (ABHD6), with an IC50 of 0.31 nM in Neuro2A cells[1]. |
| Name | KT203 |
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| Description | KT203 is a potent and selective inhibitor of α/β-hydrolase domain containing 6 (ABHD6), with an IC50 of 0.31 nM in Neuro2A cells[1]. |
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| Related Catalog | |
| Target |
IC50: 0.31 nM (ABHD6 in Neuro2A cells)[1]. |
| References |
| Molecular Formula | C28H26N4O3 |
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| Molecular Weight | 466.53 |
| Storage condition | 2-8℃ |
| RIDADR | NONH for all modes of transport |
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Discovery and optimization of piperidyl-1,2,3-triazole ureas as potent, selective, and in vivo-active inhibitors of α/β-hydrolase domain containing 6 (ABHD6).
J. Med. Chem. 56(21) , 8270-9, (2013) α/β-Hydrolase domain containing 6 (ABHD6) is a transmembrane serine hydrolase that hydrolyzes the endogenous cannabinoid 2-arachidonoylglycerol (2-AG) to regulate certain forms of cannabinoid receptor... |