Apimostinel
Modify Date: 2024-01-01 20:01:38
Apimostinel structure
|
Common Name | Apimostinel | ||
|---|---|---|---|---|
| CAS Number | 1421866-48-9 | Molecular Weight | 503.591 | |
| Density | 1.3±0.1 g/cm3 | Boiling Point | 878.7±65.0 °C at 760 mmHg | |
| Molecular Formula | C25H37N5O6 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | 485.2±34.3 °C | |
Use of ApimostinelApimostinel is an oral NMDA receptor partial agonist. |
| Name | apimostinel |
|---|---|
| Synonym | More Synonyms |
| Description | Apimostinel is an oral NMDA receptor partial agonist. |
|---|---|
| Related Catalog | |
| In Vitro | Apimostinel (NRX-1074) modulates the NMDA receptor in a similar fashion to GLYX-13, but has a synthetic modification to one of the amino acids, conferring increased potency and oral bioavailability[1]. |
| In Vivo | In preclinical models the two compounds both appear to be highly efficacious across a number of CNS disorders[1]. |
| References |
| Density | 1.3±0.1 g/cm3 |
|---|---|
| Boiling Point | 878.7±65.0 °C at 760 mmHg |
| Molecular Formula | C25H37N5O6 |
| Molecular Weight | 503.591 |
| Flash Point | 485.2±34.3 °C |
| Exact Mass | 503.274384 |
| LogP | 0.22 |
| Vapour Pressure | 0.0±0.3 mmHg at 25°C |
| Index of Refraction | 1.608 |
| Storage condition | 2-8℃ |
| NRX-1074 |
| L-Threonyl-L-prolyl-2-benzyl-L-prolyl-L-threoninamide |
| apimostinel |
| UNII:TTT1F11FZB |
| TTT1F11FZB |
| L-Threoninamide, L-threonyl-L-prolyl-2-(phenylmethyl)-L-prolyl- |