pepticinnamin E

Modify Date: 2024-01-14 19:50:43

pepticinnamin E structure	Common Name	pepticinnamin E
	CAS Number	147317-36-0	Molecular Weight	908.43400
	Density	1.284g/cm3	Boiling Point	1124.3ºC at 760 mmHg
	Molecular Formula	C₄₉H₅₄ClN₅O₁₀	Melting Point	N/A
	MSDS	N/A	Flash Point	633.7ºC

Use of pepticinnamin E

Pepticinnamin E is a Farnesyltransferase (FTase) inhibitor (IC50=42 µM). Pepticinnamin E can be used in cancer and malaria research[1][2].

Name	[(2R)-3,6-dioxopiperazin-2-yl]methyl (2R,4R)-2-benzyl-2-[[(2S)-3-(2-chloro-3-hydroxy-4-methoxyphenyl)-2-(methylamino)propanoyl]-methylamino]-5-(4-hydroxyphenyl)-3-oxo-4-[[(E)-3-[2-[(E)-pent-2-enyl]phenyl]prop-2-enoyl]amino]pentanoate
Synonym	More Synonyms

Description	Pepticinnamin E is a Farnesyltransferase (FTase) inhibitor (IC50=42 µM). Pepticinnamin E can be used in cancer and malaria research[1][2].
Related Catalog	Research Areas >> Cancer Research Areas >> Infection Signaling Pathways >> Metabolic Enzyme/Protease >> Farnesyl Transferase
Target	IC50: 42 µM (Farnesyltransferase)[1].
References	[1]. Hinterding K, et al. Synthesis and In Vitro Evaluation of the Ras Farnesyltransferase Inhibitor Pepticinnamin E. Angew Chem Int Ed Engl. 1998 May 18;37(9):1236-1239. [2]. Santa Maria KC, et al. Targeted Rediscovery and Biosynthesis of the Farnesyl-Transferase Inhibitor Pepticinnamin E. Chembiochem. 2019 Jun 3;20(11):1387-1393.

Density	1.284g/cm3
Boiling Point	1124.3ºC at 760 mmHg
Molecular Formula	C₄₉H₅₄ClN₅O₁₀
Molecular Weight	908.43400
Flash Point	633.7ºC
Exact Mass	907.35600
PSA	223.17000
LogP	5.78970
Vapour Pressure	0mmHg at 25°C
Index of Refraction	1.612

Pepticinnamin E

Pepticinnamine E

Dayang Chem (Hangzhou) Co., Ltd.
China
Product Name: pepticinnamin E
Price: $Inquiry/100g $Inquiry/1kg $Inquiry/100kg $Inquiry/1000kg
Purity: 98.0%
Delivery: Inquiry
Contact: Ms Wang
Email: enquiry@dycnchem.com

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